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25,000+
特异性抑制剂、激动剂和化合物筛选库,专注于信号通路和疾病研究领域。全球文献广泛引用,质控体系严格,100%客户满意保障。BREQUINAR (DUP785)
Brequinar (DUP785) is a potent inhibitor of dihydroorotate dehydrogenase (DHODH) with an IC50 of 5.2 nM for human DHODH. Brequinar has potent activities against a broad spectrum of viruses. In Vitro. Brequinar reduces virus progeny production by >90%, with EC 50 of 17 nM. Brequinar (5 μM) also inhibits other orthopoxviruses,and blocks virus
MQAE | DYE REAGENT | MCETRANSLATE THIS PAGE MQAE is a fluorescent indicator that is quenched via collision with chloride, and is more sensitive and selective than 36 Cl and microelectrode-based methods for chloride measurement in cells. In Vitro. Bath-applied to acute brain slices, MQAE provides high-qualityMG-132 (MG132)
MG-132 (Z-Leu-Leu-Leu-al) is a potent proteasome and calpain inhibitor with IC50 s of 100 nM and 1.2 μM, respectively. MG-132 effectively blocks the proteolytic activity of the 26S proteasome complex. MG-132, a peptide aldehyde, also is an autophagy activator . MG-132 also induces apoptosis . CL 316243 | Β3-ADRENOCEPTOR AGONIST | MCETRANSLATE THIS PAGE CL316243 is a highly potent selective β3-adrenoceptor agonist with a EC50 of 3 nM, but is an extremely poor to β1/2- receptors .CL316243 is a effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate . CL316243 has the potential for the treatment obesity, diabetes andurge urinary
NOCODAZOLE (ONCODAZOLE,诺考达唑) Nocodazole (Oncodazole) is a rapidly-reversible inhibitor of microtubule. Nocodazole binds to β-tubulin and disrupts microtubule assembly/disassembly dynamics, which prevents mitosis and induces apoptosis in tumor cells. Nocodazole inhibits Bcr-Abl, and activates CRISPR/Cas9 . IC 50 & Target. BAFILOMYCIN A1 (巴佛洛霉素A1) Bafilomycin A1 is a specific and reversible inhibitor of vacuolar H+-ATPase ( V-ATPase) with I50 values of 4-400 nmol/mg. Bafilomycin A1, a macrolide antibiotic, is also used as an autophagy inhibitor at the late stage. Bafilomycin A1 blocks autophagosome-lysosome fusion and inhibits acidification and protein degradation in lysosomes of 4-PHENYLBUTYRIC ACID (4-PBA,4-苯基丁酸) 4-Phenylbutyric acid (4-PBA) is an inhibitor of HDAC, inhibits the growth of NSCLC Cell Lines at 2 mM. Benzenebutyric acid in combination with ciglitizone results in enhanced growth arrest of cancer cells.4-Phenylbutyric acid (0-5 mM) inhibits ASFV infection in a dose-dependent manner. UPADACITINIB (ABT-494,乌帕替尼) Upadacitinib (ABT-494) 是一种高效的、具有口服活性的、选择性 Janus 激酶 1 (JAK1) 抑制剂 (IC50=43 nM)。Upadacitinib 对 JAK1 的选择性约为 JAK2 (200 nM)的 74 倍。Upadacitinib 可用于多种自身免疫性疾病的研究。- 高纯度,全球文献引用。 LY294002 | PI3K 抑制剂 | MCETRANSLATE THIS PAGE LY294002 是一种广谱 PI3K 抑制剂,抑制 PI3Kα, PI3Kδ 和 PI3Kβ 的 IC50 分别为 0.5, 0.57, 0.97 μM。LY294002 也可抑制 CK2 的活性,IC50 为 98 nM。LY294002 是一种竞争性 DNA-PK 抑制剂,可逆结合 DNA-PK 的激酶结构域,IC50 为 1.4 μM。LY294002 是一种自噬 (autophagy) 和凋亡 (apoptosis)激活剂。
MCE-您身边的抑制剂大师 MCE (MedChemExpress) 为生命科学和医药研发人员提供25,000+
特异性抑制剂、激动剂和化合物筛选库,专注于信号通路和疾病研究领域。全球文献广泛引用,质控体系严格,100%客户满意保障。BREQUINAR (DUP785)
Brequinar (DUP785) is a potent inhibitor of dihydroorotate dehydrogenase (DHODH) with an IC50 of 5.2 nM for human DHODH. Brequinar has potent activities against a broad spectrum of viruses. In Vitro. Brequinar reduces virus progeny production by >90%, with EC 50 of 17 nM. Brequinar (5 μM) also inhibits other orthopoxviruses,and blocks virus
MQAE | DYE REAGENT | MCETRANSLATE THIS PAGE MQAE is a fluorescent indicator that is quenched via collision with chloride, and is more sensitive and selective than 36 Cl and microelectrode-based methods for chloride measurement in cells. In Vitro. Bath-applied to acute brain slices, MQAE provides high-qualityMG-132 (MG132)
MG-132 (Z-Leu-Leu-Leu-al) is a potent proteasome and calpain inhibitor with IC50 s of 100 nM and 1.2 μM, respectively. MG-132 effectively blocks the proteolytic activity of the 26S proteasome complex. MG-132, a peptide aldehyde, also is an autophagy activator . MG-132 also induces apoptosis . CL 316243 | Β3-ADRENOCEPTOR AGONIST | MCETRANSLATE THIS PAGE CL316243 is a highly potent selective β3-adrenoceptor agonist with a EC50 of 3 nM, but is an extremely poor to β1/2- receptors .CL316243 is a effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate . CL316243 has the potential for the treatment obesity, diabetes andurge urinary
NOCODAZOLE (ONCODAZOLE,诺考达唑) Nocodazole (Oncodazole) is a rapidly-reversible inhibitor of microtubule. Nocodazole binds to β-tubulin and disrupts microtubule assembly/disassembly dynamics, which prevents mitosis and induces apoptosis in tumor cells. Nocodazole inhibits Bcr-Abl, and activates CRISPR/Cas9 . IC 50 & Target. BAFILOMYCIN A1 (巴佛洛霉素A1) Bafilomycin A1 is a specific and reversible inhibitor of vacuolar H+-ATPase ( V-ATPase) with I50 values of 4-400 nmol/mg. Bafilomycin A1, a macrolide antibiotic, is also used as an autophagy inhibitor at the late stage. Bafilomycin A1 blocks autophagosome-lysosome fusion and inhibits acidification and protein degradation in lysosomes of 4-PHENYLBUTYRIC ACID (4-PBA,4-苯基丁酸) 4-Phenylbutyric acid (4-PBA) is an inhibitor of HDAC, inhibits the growth of NSCLC Cell Lines at 2 mM. Benzenebutyric acid in combination with ciglitizone results in enhanced growth arrest of cancer cells.4-Phenylbutyric acid (0-5 mM) inhibits ASFV infection in a dose-dependent manner. UPADACITINIB (ABT-494,乌帕替尼) Upadacitinib (ABT-494) 是一种高效的、具有口服活性的、选择性 Janus 激酶 1 (JAK1) 抑制剂 (IC50=43 nM)。Upadacitinib 对 JAK1 的选择性约为 JAK2 (200 nM)的 74 倍。Upadacitinib 可用于多种自身免疫性疾病的研究。- 高纯度,全球文献引用。 LY294002 | PI3K 抑制剂 | MCETRANSLATE THIS PAGE LY294002 是一种广谱 PI3K 抑制剂,抑制 PI3Kα, PI3Kδ 和 PI3Kβ 的 IC50 分别为 0.5, 0.57, 0.97 μM。LY294002 也可抑制 CK2 的活性,IC50 为 98 nM。LY294002 是一种竞争性 DNA-PK 抑制剂,可逆结合 DNA-PK 的激酶结构域,IC50 为 1.4 μM。LY294002 是一种自噬 (autophagy) 和凋亡 (apoptosis)激活剂。
RESIQUIMOD (R848,雷西莫特) Resiquimod is a Toll-like receptor 7 and 8 ( TLR7/TLR8) agonist that induces the upregulation of cytokines such as TNF-α, IL-6 and IFN-α. IC 50 & Target. TLR7/TLR8. In Vitro. Resiquimod (R-848) induces both hapten- and allergen-specific circulating T cells, including TH2 effectors, to produce IFN-γ and even to lose the ability to produceIL
VCMMAE (MC-VC-PAB-MMAE) VcMMAE (mc-vc-PAB-MMAE) is a drug-linker conjugate for ADC with potent antitumor activity by using the anti-mitotic agent, monomethyl auristatin E (MMAE, a tubulin inhibitor), linked via the lysosomally cleavable dipeptide, valine-citrulline (vc). IC 50 & Target. Auristatin. In Vitro. Monomethyl auristatin E (MMAE) is efficientlyreleased from
U-73122 | PHOSPHOLIPASE C 抑制剂 | MCE U-73122 is a phospholipase C (PLC) and 5-LO (5-lipoxygenase) inhibitor with an IC50 of 1-2.1 µM for PLC. IC 50 & Target. 5-LOX. In Vitro. U-73122 potently inhibits receptor-coupled activation of PLC in membranes isolated from PMNs . U-73122 inhibits N-formyl-methionyl-leucyl-phenylalanine-induced aggregation of humanpolymorphonuclear
MQAE | DYE REAGENT | MCETRANSLATE THIS PAGE MQAE is a fluorescent indicator that is quenched via collision with chloride, and is more sensitive and selective than 36 Cl and microelectrode-based methods for chloride measurement in cells. In Vitro. Bath-applied to acute brain slices, MQAE provides high-quality 4-PHENYLBUTYRIC ACID (4-PBA,4-苯基丁酸) 4-Phenylbutyric acid (4-PBA) is an inhibitor of HDAC, inhibits the growth of NSCLC Cell Lines at 2 mM. Benzenebutyric acid in combination with ciglitizone results in enhanced growth arrest of cancer cells.4-Phenylbutyric acid (0-5 mM) inhibits ASFV infection in a dose-dependent manner. BORTEZOMIB (PS-341,硼替佐米) Bortezomib (PS-341) 是一种可逆性和选择性的蛋白酶体 (proteasome) 抑制剂,通过靶向苏氨酸残基有效抑制 20S 蛋白酶体 (Ki=0.6 nM)。Bortezomib 破坏细胞周期、诱导细胞凋亡以及抑制核因子NF-κB。Bortezomib
是第一种蛋白酶体抑制剂,具有抗癌活性。- 高纯度,全球文献引用。 UPADACITINIB (ABT-494,乌帕替尼) Upadacitinib (ABT-494) 是一种高效的、具有口服活性的、选择性 Janus 激酶 1 (JAK1) 抑制剂 (IC50=43 nM)。Upadacitinib 对 JAK1 的选择性约为 JAK2 (200 nM)的 74 倍。Upadacitinib 可用于多种自身免疫性疾病的研究。- 高纯度,全球文献引用。 BAFILOMYCIN A1 (巴佛洛霉素A1) Bafilomycin A1 是特异性,可逆的 V-ATPase 抑制剂,I50 值为 4-400 nmol/mg。Bafilomycin A1,大环内酯类抗生素, 是一种自噬 (autophagy) 晚期阶段抑制剂。Bafilomycin A1 阻断自噬体与溶酶体的融合,并抑制培养细胞溶酶体中的酸化和蛋白质降解。Bafilomycin A1 也诱导调亡 (apoptosis)。 CYTOCHALASIN D (ZYGOSPORIN A,细胞松弛素D) Cytochalasin D (Zygosporin A; NSC 209835) 是一种有效、细胞渗透性的肌动蛋白聚合抑制剂,由真菌产生,通过绑定 G-actin 抑制 G-actin–cofilin 的相互作用。Cytochalasin D 还能抑制 cofilin 与 F-actin 的结合,降低了活细胞中肌动蛋白聚合和解聚的速率。Cytochalasin D 可以减少外泌体的释放,进而减少肿瘤环境中survivin
Y-27632 | SELECTIVE ROCK 抑制剂 | MCETRANSLATE THIS PAGE Y-27632 是口服有效的, ATP 竞争性的 ROCK-I 和 ROCK-II 抑制剂,Ki 分别为 220 nM 和 300 nM。Y-27632 诱导凋亡 (apoptosis)。Y-27632 通过上皮-间充质过渡样调节引发人诱导多能干细胞 (hIPSCs) 选择性地分化为间胚层谱系。- 高纯度,全球文献引用。 — MASTER OF SMALL MOLECULES "暑" 于我的 "夏" 午茶 致电400-820-3792或联系在线客服Cart (0)
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研究领域
*
天然产物
*
客户验证
* •Anti-infection
* •Antibody-drug Conjugate/ADC Related* •Apoptosis
* •Autophagy
* •Cell Cycle/DNA Damage* •Cytoskeleton
* •Epigenetics
* •GPCR/G Protein
* •Immunology/Inflammation * •JAK/STAT Signaling * •MAPK/ERK Pathway * •Membrane Transporter/Ion Channel * •Metabolic Enzyme/Protease * •Neuronal Signaling* •NF-κB
* •PI3K/Akt/mTOR
* •PROTAC
* •Protein Tyrosine Kinase/RTK* •Stem Cell/Wnt
* •TGF-beta/Smad
* •Vitamin D Related* •Others
* •Cancer
* •Cardiovascular Disease* •Endocrinology
* •Infection
* •Inflammation/Immunology * •Metabolic Disease * •Neurological Disease* •Others
* •Saccharides and Glycosides * •Phenylpropanoids* •Quinones
* •Flavonoids
* •Terpenoids and Glycosides* •Steroids
* •Alkaloid
* •Phenols
* •Acids and Aldehydes* •Others
*
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